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BG31227A4 - Метод за получаване на рацемични или оптично активни пирамидо (1,2 а)хетероциклични съединения - Google Patents

Метод за получаване на рацемични или оптично активни пирамидо (1,2 а)хетероциклични съединения

Info

Publication number
BG31227A4
BG31227A4 BG036221A BG3622176A BG31227A4 BG 31227 A4 BG31227 A4 BG 31227A4 BG 036221 A BG036221 A BG 036221A BG 3622176 A BG3622176 A BG 3622176A BG 31227 A4 BG31227 A4 BG 31227A4
Authority
BG
Bulgaria
Prior art keywords
racemic
pjromido
oropticallj
heterocjlic
commpounds
Prior art date
Application number
BG036221A
Other languages
English (en)
Inventor
Zoltan Meszaros
Jozef Knoll
Peter Szentmiklosi
Istvan Hermecz
Agnes Horvath
Sandor Virag
Lelle Vasvari
Agoston David
Original Assignee
Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt. filed Critical Chinoin Gyogyszer Es Vegyeszeti Termekek Gyara Rt.
Publication of BG31227A4 publication Critical patent/BG31227A4/bg

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P7/00—Drugs for disorders of the blood or the extracellular fluid
    • A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pain & Pain Management (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Rheumatology (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Plural Heterocyclic Compounds (AREA)

Abstract

Метод за получаване на охарактеризирани и доказани в описанието рацемични или оптически активни пиримидо-(1,2а) хетероциклични съединения с обща формула................................ Патентните претенции са формулирани в 4 точки
BG036221A 1975-11-27 1976-11-16 Метод за получаване на рацемични или оптично активни пирамидо (1,2 а)хетероциклични съединения BG31227A4 (bg)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
HU75CI1623A HU173438B (hu) 1975-11-27 1975-11-27 Sposob poluchenija novykh proizvodnykh 4-okso-1,6,7,8-/tetragidro-4h-pirido/1,2/pirimidina s zaderzhivajuhhejj vozgoranie aktivnot'ju i protivosvertivajuhhem effektom

Publications (1)

Publication Number Publication Date
BG31227A4 true BG31227A4 (bg) 1981-11-16

Family

ID=10994587

Family Applications (1)

Application Number Title Priority Date Filing Date
BG036221A BG31227A4 (bg) 1975-11-27 1976-11-16 Метод за получаване на рацемични или оптично активни пирамидо (1,2 а)хетероциклични съединения

Country Status (28)

Country Link
US (2) US4460771A (bg)
JP (1) JPS5914033B2 (bg)
AT (1) AT359506B (bg)
AU (1) AU512256B2 (bg)
BE (1) BE848868A (bg)
BG (1) BG31227A4 (bg)
CA (1) CA1088531A (bg)
CH (2) CH630378A5 (bg)
CS (1) CS203135B2 (bg)
DD (1) DD130431A5 (bg)
DE (1) DE2653257A1 (bg)
DK (1) DK153150C (bg)
EG (1) EG12495A (bg)
ES (1) ES453690A1 (bg)
FI (1) FI62085C (bg)
FR (1) FR2332755A1 (bg)
GB (1) GB1531963A (bg)
GR (1) GR61820B (bg)
HU (1) HU173438B (bg)
IL (1) IL50930A (bg)
IN (1) IN148945B (bg)
MX (1) MX5178E (bg)
NL (1) NL188948C (bg)
PL (1) PL109657B1 (bg)
RO (2) RO79705A (bg)
SE (1) SE433353B (bg)
SU (2) SU664565A3 (bg)
YU (2) YU289076A (bg)

Families Citing this family (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
HU180701B (en) * 1977-12-29 1983-04-29 Chinoin Gyogyszer Es Vegyeszet Process for preparing pyrido-/1,2-a/pyrimidines containing a carboxylic or ester group on the pirimidimering
US4192944A (en) * 1978-04-03 1980-03-11 Bristol-Myers Company Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents
US4342870A (en) * 1980-03-28 1982-08-03 Janssen Pharmaceutica N.V. Novel 3-(1-piperidinylalkyl)-4H-pyrido[1,2-a]pyrimidin-4-one derivatives
HU183408B (en) * 1981-04-28 1984-05-28 Chinoin Gyogyszer Es Vegyeszet Process for producing oral ratard pharmaceutical compositions
HU186607B (en) * 1982-03-31 1985-08-28 Chinoin Gyogyszer Es Vegyeszet Process for preparing pharmaceutical composition with synergetic antiinflammatory activity
NO162019C (no) * 1983-11-23 1989-10-25 Fujisawa Pharmaceutical Co Analogifremgangsmaate for fremstilling av terapeutisk aktive pyrimidoiskinolinderivater.
US4772475A (en) * 1985-03-08 1988-09-20 Yamanouchi Pharmaceutical Co., Ltd. Controlled-release multiple units pharmaceutical formulation
HU201551B (en) * 1988-02-03 1990-11-28 Chinoin Gyogyszer Es Vegyeszet Process for producing 4-oxo-4h-pyrido(1,2-a)pyrimidine-3-carboxylic acid amide derivatives and pharmaceutical compositions comprising same
US5252572A (en) * 1988-02-03 1993-10-12 Chinoin Gyogyszer- Es Vegyeszeti Termekek Gyara Rt. Pyridopyrimidine derivatives, pharmaceutical compositions containing them and process for preparing same
MY125533A (en) 1999-12-06 2006-08-30 Bristol Myers Squibb Co Heterocyclic dihydropyrimidine compounds
ES2278197T3 (es) * 2002-07-09 2007-08-01 Actelion Pharmaceuticals Ltd. Derivados de 7,8,9,10-tetrahidro-6h-azepino, 6,7,8,9-tetrahidro-pirido y 2,3-dihidro-2h-pirrolo(1,2-b)-quinazolinona.
US7772232B2 (en) * 2004-04-15 2010-08-10 Bristol-Myers Squibb Company Quinazolinyl compounds as inhibitors of potassium channel function
GB2423928B (en) * 2004-11-16 2008-04-09 Efflux Technology Inc Methods and compositions for treating pain

Family Cites Families (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
CH538494A (de) * 1966-11-02 1973-06-30 Chinoin Gyogyszer Es Vegyeszet Verfahren zur Herstellung neuer Homopyrimidazol-Derivate
US3642797A (en) * 1968-06-10 1972-02-15 Sterling Drug Inc 4h-pyrido(1 2-a)pyrimidin-4-ones
US4209622A (en) * 1973-03-30 1980-06-24 Chinoin Gygyszer es Vegyeszeti Termekek Gyara Rt. 3-(Ethoxycarbonyl-methyl)-6-methyl-4-oxo-6,7,8,9-tetrahydro-4H-pyrido[1,2-a]pyrimidine
HU168014B (bg) * 1973-03-30 1976-02-28
HU168541B (bg) * 1973-11-24 1976-05-28
US4022897A (en) * 1974-03-04 1977-05-10 E. R. Squibb & Sons, Inc. CNS active compounds
US3960863A (en) * 1974-06-25 1976-06-01 Sankyo Company Limited Pyrido[1,2-a]pyrimidinone derivatives
US4066766A (en) * 1975-03-03 1978-01-03 Pfizer Inc. 1-Oxo-6-substituted pyrimido [1,2-a]quinoline-2-carboxylic acids and derivatives thereof and their use as antiallergy agents
HU174693B (hu) * 1976-02-12 1980-03-28 Chinoin Gyogyszer Es Vegyeszet Sposob poluchenija kondensirovannykh proizvodnykh pirimidina
US4122274A (en) * 1977-05-25 1978-10-24 Bristol-Myers Company 3-Tetrazolo-5,6,7,8-substituted-pyrido[1,2-a]pyrimidin-4-ones
US4192944A (en) * 1978-04-03 1980-03-11 Bristol-Myers Company Optionally substituted 4-oxo-4H-pyrido[1,2-a]pyrimidine-3-N-(1H-tetrazol-4-yl)carboxamides and their use as antiallergy agents

Also Published As

Publication number Publication date
NL7613140A (nl) 1977-06-01
CS203135B2 (en) 1981-02-27
NL188948B (nl) 1992-06-16
ATA873576A (de) 1980-04-15
FI763401A (bg) 1977-05-28
IN148945B (bg) 1981-07-25
DK153150C (da) 1988-10-24
RO73522A (ro) 1981-11-04
NL188948C (nl) 1992-11-16
US4460771A (en) 1984-07-17
CH630378A5 (de) 1982-06-15
SE7613140L (sv) 1977-05-28
AT359506B (de) 1980-11-10
MX5178E (es) 1983-04-20
FR2332755A1 (fr) 1977-06-24
PL109657B1 (en) 1980-06-30
EG12495A (en) 1980-12-31
JPS5914033B2 (ja) 1984-04-02
FI62085B (fi) 1982-07-30
ES453690A1 (es) 1977-12-01
GB1531963A (en) 1978-11-15
IL50930A (en) 1981-06-29
GR61820B (en) 1979-01-22
YU147583A (en) 1986-06-30
YU289076A (en) 1983-12-31
BE848868A (fr) 1977-03-16
DE2653257C2 (bg) 1989-04-20
CH630379A5 (de) 1982-06-15
AU1975976A (en) 1978-05-25
FR2332755B1 (bg) 1978-12-22
CA1088531A (en) 1980-10-28
DK534076A (da) 1977-05-28
DD130431A5 (de) 1978-03-29
SU664565A3 (ru) 1979-05-25
DK153150B (da) 1988-06-20
DE2653257A1 (de) 1977-06-02
IL50930A0 (en) 1977-01-31
SU698532A3 (ru) 1979-11-15
HU173438B (hu) 1979-05-28
SE433353B (sv) 1984-05-21
RO79705A (ro) 1982-08-17
AU512256B2 (en) 1980-10-02
JPS5268198A (en) 1977-06-06
US4472398A (en) 1984-09-18
FI62085C (fi) 1982-11-10

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