ATE399779T1 - Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugaten - Google Patents
Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugatenInfo
- Publication number
- ATE399779T1 ATE399779T1 AT02759906T AT02759906T ATE399779T1 AT E399779 T1 ATE399779 T1 AT E399779T1 AT 02759906 T AT02759906 T AT 02759906T AT 02759906 T AT02759906 T AT 02759906T AT E399779 T1 ATE399779 T1 AT E399779T1
- Authority
- AT
- Austria
- Prior art keywords
- sub
- neuraminidase
- production
- intermediate products
- inhibitor conjugates
- Prior art date
Links
- 229940123424 Neuraminidase inhibitor Drugs 0.000 title abstract 2
- 238000004519 manufacturing process Methods 0.000 title abstract 2
- 239000002911 sialidase inhibitor Substances 0.000 title abstract 2
- 239000013067 intermediate product Substances 0.000 title 1
- 150000000180 1,2-diols Chemical class 0.000 abstract 1
- 125000006242 amine protecting group Chemical group 0.000 abstract 1
- 125000006244 carboxylic acid protecting group Chemical group 0.000 abstract 1
- 150000001875 compounds Chemical class 0.000 abstract 1
- 238000000034 method Methods 0.000 abstract 1
- 125000006239 protecting group Chemical group 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D407/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00
- C07D407/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings
- C07D407/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having oxygen atoms as the only ring hetero atoms, not provided for by group C07D405/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/12—Antivirals
- A61P31/14—Antivirals for RNA viruses
- A61P31/16—Antivirals for RNA viruses for influenza or rhinoviruses
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D309/00—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings
- C07D309/16—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
- C07D309/28—Heterocyclic compounds containing six-membered rings having one oxygen atom as the only ring hetero atom, not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
-
- Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
- Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
- Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
- Y02P20/00—Technologies relating to chemical industry
- Y02P20/50—Improvements relating to the production of bulk chemicals
- Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups
Landscapes
- Organic Chemistry (AREA)
- Chemical & Material Sciences (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Virology (AREA)
- Oncology (AREA)
- Public Health (AREA)
- Molecular Biology (AREA)
- Chemical Kinetics & Catalysis (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Pulmonology (AREA)
- Pharmacology & Pharmacy (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Communicable Diseases (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Plural Heterocyclic Compounds (AREA)
- Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
- Medicines Containing Plant Substances (AREA)
- Preparation Of Compounds By Using Micro-Organisms (AREA)
- Pyrane Compounds (AREA)
- Saccharide Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| AUPR757401 | 2001-09-07 |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| ATE399779T1 true ATE399779T1 (de) | 2008-07-15 |
Family
ID=3831510
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| AT02759906T ATE399779T1 (de) | 2001-09-07 | 2002-08-30 | Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugaten |
Country Status (12)
| Country | Link |
|---|---|
| US (1) | US7230114B2 (de) |
| EP (1) | EP1423385B1 (de) |
| JP (1) | JP4463553B2 (de) |
| AT (1) | ATE399779T1 (de) |
| BR (1) | BR0212261A (de) |
| CA (1) | CA2456239C (de) |
| DE (1) | DE60227386D1 (de) |
| DK (1) | DK1423385T3 (de) |
| ES (1) | ES2307776T3 (de) |
| MX (1) | MXPA04002141A (de) |
| PT (1) | PT1423385E (de) |
| WO (1) | WO2003022841A1 (de) |
Families Citing this family (2)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2015032357A1 (zh) * | 2013-09-09 | 2015-03-12 | 中国科学院上海有机化学研究所 | 扎那米韦和拉那米韦的中间体及其合成方法 |
| CN113461631B (zh) * | 2021-06-29 | 2022-10-14 | 上海应用技术大学 | 一种1,3,4-恶二唑类神经氨酸酶抑制剂及其制备方法与应用 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| GB9516276D0 (en) | 1995-08-08 | 1995-10-11 | Biota Scient Management | Chemical compounds |
| DE69721242T2 (de) | 1996-03-01 | 2004-01-29 | Biota Scient Management | Verfahren zum nachweis von influenza-virus und dazu verwendbare verbindungen |
| CA2263336C (en) * | 1996-08-13 | 2007-03-13 | Sankyo Company, Limited | Neuraminic acid compounds |
| AUPR001000A0 (en) * | 2000-09-08 | 2000-10-05 | Biota Scientific Management Pty Ltd | Novel chemical compounds and their use |
-
2002
- 2002-08-30 EP EP02759906A patent/EP1423385B1/de not_active Expired - Lifetime
- 2002-08-30 US US10/488,791 patent/US7230114B2/en not_active Expired - Fee Related
- 2002-08-30 CA CA2456239A patent/CA2456239C/en not_active Expired - Fee Related
- 2002-08-30 MX MXPA04002141A patent/MXPA04002141A/es active IP Right Grant
- 2002-08-30 WO PCT/AU2002/001187 patent/WO2003022841A1/en active IP Right Grant
- 2002-08-30 AT AT02759906T patent/ATE399779T1/de not_active IP Right Cessation
- 2002-08-30 DE DE60227386T patent/DE60227386D1/de not_active Expired - Lifetime
- 2002-08-30 BR BR0212261-8A patent/BR0212261A/pt not_active IP Right Cessation
- 2002-08-30 PT PT02759906T patent/PT1423385E/pt unknown
- 2002-08-30 ES ES02759906T patent/ES2307776T3/es not_active Expired - Lifetime
- 2002-08-30 DK DK02759906T patent/DK1423385T3/da active
- 2002-08-30 JP JP2003526916A patent/JP4463553B2/ja not_active Expired - Fee Related
Also Published As
| Publication number | Publication date |
|---|---|
| PT1423385E (pt) | 2008-09-24 |
| JP4463553B2 (ja) | 2010-05-19 |
| ES2307776T3 (es) | 2008-12-01 |
| BR0212261A (pt) | 2004-10-19 |
| CA2456239A1 (en) | 2003-03-20 |
| WO2003022841A1 (en) | 2003-03-20 |
| MXPA04002141A (es) | 2004-07-23 |
| EP1423385A1 (de) | 2004-06-02 |
| CA2456239C (en) | 2010-11-30 |
| DK1423385T3 (da) | 2008-11-03 |
| US20050032853A1 (en) | 2005-02-10 |
| JP2005501921A (ja) | 2005-01-20 |
| EP1423385B1 (de) | 2008-07-02 |
| US7230114B2 (en) | 2007-06-12 |
| EP1423385A4 (de) | 2004-12-01 |
| DE60227386D1 (de) | 2008-08-14 |
Similar Documents
| Publication | Publication Date | Title |
|---|---|---|
| NO20062644L (no) | DPP-IV inhibitorer | |
| PL369740A1 (en) | Novel dihydropteridinones, method for producing the same and the use thereof as medicaments | |
| MEP43408A (en) | Novel fluorene carboxylic acid esters, methods for the production thereof, and use of the same as pharmaceuticals | |
| BR0307432A (pt) | Difluormetiltiazolilcarboxanilidas | |
| TR200201168T2 (tr) | CGRP-Antagonistleri-yeni siklopropanlar içeren ilaçlar ve üretim yöntemleri. | |
| SE0004245D0 (sv) | Novel compounds and their use | |
| ATE288900T1 (de) | Substituierte benzoylcyclohexandione | |
| BRPI0410861A (pt) | métodos e composições para a produção de aminoácidos | |
| MXPA03009548A (es) | Arilsulfonamidas como agentes antivirales. | |
| DE60221508D1 (de) | Aminosäurederivate als hiv-protease-inhibitoren | |
| TR28332A (tr) | Arilasetik asit türevleri. | |
| DE50310579D1 (de) | Furancarboxamide | |
| BR0316549A (pt) | ésteres de ácido carbamìnico com efeito anticolinérgico | |
| WO2001090102A3 (de) | 6-heterocyclyl-3-oxo-3,4-dihydro-chinoxaline | |
| WO2002088125A3 (de) | Triazolopyrimidine mit fungizider wirkung | |
| DE50311756D1 (de) | Mikrobizide oxathiincarboxamide | |
| ATE399779T1 (de) | Zwischenprodukte für die herstellung von neuraminidase-inhibitor-konjugaten | |
| BR0013751A (pt) | Processo para produção de derivados de ácido naftiridina-3-carboxìlico | |
| DK1347965T3 (da) | Hidtil ukendte desloratidinsalte, fremgangsmåde til syntese deraf samt farmaceutiske præparater deraf | |
| MXPA02001406A (es) | Heterociclilos-2h-cromenos substituidos. | |
| DE60112241D1 (de) | Verfahren und zwischenverbindungen zur herstellung von imidazopyridinen | |
| FR2823503B1 (fr) | Nouveaux composes, procede de fabrication, utilisation comme pigments et composition cosmetique | |
| EP1479667A4 (de) | Verfahren zur herstellung einer chromonverbindung | |
| CA2425164A1 (en) | (4-acylaminopiperidin-1-yl)acetamides as neurokinin antagonists | |
| WO2001010862A3 (de) | Substituierte heterocyclylbenzofurane |
Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| RER | Ceased as to paragraph 5 lit. 3 law introducing patent treaties |