Abstract
Among the diverse co-regulatory relationships between transcription factors (TFs) and microRNAs (miRNAs), feedback loops have received the most extensive research attention. The co-regulation of TFs and miRNAs plays an important role in colorectal cancer (CRC) growth. Here, we show that miR-124 can regulate two isoforms of p63, TAp63 and ΔNp63, via iASPP, while p63 modulates signal transducers and activators of transcription 1 (STAT1) expression by targeting miR-155. Moreover, STAT1 acts as a regulator of CRC growth by targeting miR-124. Taken together, these results reveal a feedback loop between miRNAs and TFs. This feedback loop comprises miR-124, iASPP, STAT1, miR-155, TAp63 and ΔNp63, which are essential for CRC growth. Moreover, this feedback loop is perturbed in human colon carcinomas, which suggests that the manipulation of this microRNA-TF feedback loop has therapeutic potential for CRC.
Keywords:
cell growth; colorectal cancer; feedback loop; miR-124; p63.
MeSH terms
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Animals
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Cell Line, Tumor
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Cell Proliferation
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Chromatin Immunoprecipitation
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Colorectal Neoplasms / genetics*
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Colorectal Neoplasms / pathology
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Feedback, Physiological*
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Female
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Gene Expression Regulation, Neoplastic*
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Gene Knockdown Techniques
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Humans
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Intracellular Signaling Peptides and Proteins / genetics
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Intracellular Signaling Peptides and Proteins / metabolism*
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Mice
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Mice, Inbred BALB C
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Mice, Nude
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MicroRNAs / genetics
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MicroRNAs / metabolism*
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Protein Isoforms / metabolism
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RNA Interference
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RNA, Small Interfering / metabolism
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Repressor Proteins / genetics
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Repressor Proteins / metabolism*
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STAT1 Transcription Factor / genetics
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STAT1 Transcription Factor / metabolism
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Signal Transduction
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Transcription Factors / genetics*
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Transcription Factors / metabolism
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Tumor Suppressor Proteins / genetics*
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Tumor Suppressor Proteins / metabolism
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Xenograft Model Antitumor Assays
Substances
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Intracellular Signaling Peptides and Proteins
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MIRN124 microRNA, human
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MIRN155 microRNA, human
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MicroRNAs
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PPP1R13L protein, human
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Protein Isoforms
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RNA, Small Interfering
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Repressor Proteins
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STAT1 Transcription Factor
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STAT1 protein, human
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TP63 protein, human
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Transcription Factors
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Tumor Suppressor Proteins